Location via proxy:   [ UP ]  
[Report a bug]   [Manage cookies]                

Quercetin attenuates oxygen-glucose deprivation- and excitotoxin-induced neurotoxicity in primary cortical cell cultures

Biol Pharm Bull. 2003 Apr;26(4):544-6. doi: 10.1248/bpb.26.544.

Abstract

The possible role of quercetin, a naturally occurring plant flavonoid, in protecting against oxygen-glucose deprivation (OGD)-, excitotoxins-, and free radical-induced neuronal injury in mouse cortical cell cultures was investigated. Pre- and co-treatment with quercetin (100 microM) inhibited 50 min OGD-, 20 microM N-methyl-D-aspartate (NMDA)-, and 50 microM kainate-induced neurotoxicity by 36, 22, and 61%, respectively. Quercetin significantly ameliorated free radical-induced neuronal injury caused by buthionine sulfoximine, sodium nitroprusside, ZnCl(2), and FeCl(2). These results suggest that quercetin may contribute a neuroprotective action against ischemic neural injury, partially via antioxidant actions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Cell Hypoxia / drug effects
  • Cell Hypoxia / physiology
  • Cells, Cultured
  • Cerebral Cortex / drug effects*
  • Cerebral Cortex / pathology
  • Cerebral Cortex / physiology
  • Dose-Response Relationship, Drug
  • Excitatory Amino Acid Agonists / toxicity*
  • Glucose / deficiency*
  • Kainic Acid / toxicity
  • Mice
  • Mice, Inbred ICR
  • N-Methylaspartate / toxicity
  • Neuroglia / drug effects
  • Neuroglia / pathology
  • Neuroglia / physiology
  • Neurons / drug effects
  • Neurons / pathology
  • Neurons / physiology
  • Oxygen / metabolism*
  • Quercetin / pharmacology*

Substances

  • Antioxidants
  • Excitatory Amino Acid Agonists
  • N-Methylaspartate
  • Quercetin
  • Glucose
  • Oxygen
  • Kainic Acid