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Physiological effects of 4-aminopyridine on demyelinated mammalian motor and sensory fibers

Ann Neurol. 1987 Aug;22(2):264-8. doi: 10.1002/ana.410220212.

Abstract

The selective response of demyelinated sensory fibers to 4-aminopyridine (4-AP) has been proposed as a mechanism underlying the reported paresthesias that complicate the use of this potassium-channel blocking agent in clinical trials for the treatment of multiple sclerosis and neuromuscular disorders. To identify differences in the electrophysiological response of specific fiber types to the application of 4-AP, rat ventral and dorsal spinal roots, demyelinated by intrathecal injections of lysophosphatidylcholine, were examined in vitro before and during potassium-channel blockade. The compound action potentials of demyelinated ventral roots showed a prominent postspike negativity associated with a broadening of single action potentials following application of 4-AP. Under similar conditions, whole root responses of demyelinated dorsal root axons also developed a late negativity, but individual fibers were observed to fire repetitively in response to a single stimulus. The data support the hypothesis that the prominent sensory dysfunctions reported in clinical trials of 4-AP are due to the selective response characteristics of sensory fibers.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 4-Aminopyridine
  • Action Potentials
  • Aminopyridines / pharmacology*
  • Animals
  • Axons / drug effects
  • Axons / physiology
  • Female
  • Lysophosphatidylcholines / pharmacology*
  • Motor Activity / physiology*
  • Myelin Sheath / drug effects*
  • Nerve Fibers, Myelinated / drug effects*
  • Nerve Fibers, Myelinated / physiology
  • Rats
  • Sensation / physiology*
  • Spinal Nerve Roots / drug effects
  • Spinal Nerve Roots / physiology

Substances

  • Aminopyridines
  • Lysophosphatidylcholines
  • 4-Aminopyridine