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scholarly journals A Recent Overview of 1,2,3-Triazole-Containing Hybrids as Novel Antifungal Agents: Focusing on Synthesis, Mechanism of Action, and Structure-Activity Relationship (SAR)

2022 ◽  
Vol 2022 ◽  
pp. 1-50
Author(s):  
Mahrokh Marzi ◽  
Mojtaba Farjam ◽  
Zahra Kazeminejad ◽  
Abolfazl Shiroudi ◽  
Amin Kouhpayeh ◽  
...  

A pharmacophore system has been found as 1,2,3-triazole, a five-membered heterocycle ring with nitrogen heteroatoms. These heterocyclic compounds can be produced using azide-alkyne cycloaddition processes catalyzed by ruthenium or copper. The bioactive compounds demonstrated antitubercular, antibacterial, anti-inflammatory, anticancer, antioxidant, antiviral, and antidiabetic properties. This heterocycle molecule, in particular, with one or more 1,2,3-triazole cores has been found to have the most powerful antifungal effects. The goal of this review is to highlight recent developments in the synthesis and structure-activity relationship (SAR) investigation of this prospective fungicidal chemical. Also there have been explained drugs and mechanism of action of a triazole compound with antifungal activity. This review will be useful in a variety of fields, including medicinal chemistry, organic chemistry, mycology, and pharmacology.

Author(s):  
Giovanny Carvalho dos Santos ◽  
Lucas Michelão Martins ◽  
Bruna Andressa Bregadiolli ◽  
Vitor Fernandes Moreno ◽  
Luiz Carlos da Silva‐Filho ◽  
...  

2018 ◽  
Vol 38 (2) ◽  
pp. 49-76 ◽  
Author(s):  
Amna Kamal ◽  
Muhammad Adnan Iqbal ◽  
Haq Nawaz Bhatti

AbstractSelenium is a biocompatible element and participates in several biochemical reactions occurring in the human body. Its biocompatibility and minimal toxicity has attracted researchers to develop selenium-based drugs. Hence, recent developments on biomedical applications of selenium-based compounds have been discussed. A structure activity relationship has also been interpreted.


MedChemComm ◽  
2011 ◽  
Vol 2 (8) ◽  
pp. 689-697 ◽  
Author(s):  
Daniel Pla ◽  
Fernando Albericio ◽  
Mercedes Álvarez

The latest developments towards the synthesis of lamellarins, their structure–activity relationship and advances in the mechanism of action are described.


2014 ◽  
Vol 3 (2) ◽  
pp. 117-126 ◽  
Author(s):  
Ganesh Samala ◽  
Shruti Singh Kakan ◽  
Radhika Nallangi ◽  
Parthiban Brindha Devi ◽  
Jonnalagadda Padma Sridevi ◽  
...  

2013 ◽  
Vol 27 (11) ◽  
pp. 951-964 ◽  
Author(s):  
El Hassane Anouar ◽  
Salwa Raweh ◽  
Imene Bayach ◽  
Muhammad Taha ◽  
Mohd Syukri Baharudin ◽  
...  

2010 ◽  
Vol 53 (1) ◽  
pp. 61-76 ◽  
Author(s):  
Jiangnan Peng ◽  
Sucheta Kudrimoti ◽  
Sivaprakasam Prasanna ◽  
Srinivas Odde ◽  
Robert J. Doerksen ◽  
...  

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