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- إيثيل فينيدات هو منبّه ومشابه بنيوي قريب من ميثيل فينيدات. تقوم هذه المادة بدور مثبط استرداد للدوبامين وللنورإبينفرين، مما يرفع من تركيز هذه النواقل العصبية في الدماغ. يستقلب إيثيل فينيدات إلى ميثيل فينيدات ، وتتم العملية في الكبد عبر تفاعل . (ar)
- Ethylphenidate (EPH), also known as Baxtercaine in the United Kingdom is a psychostimulant and a close analog of methylphenidate. Ethylphenidate acts as both a dopamine reuptake inhibitor and norepinephrine reuptake inhibitor, meaning it effectively boosts the levels of the norepinephrine and dopamine neurotransmitters in the brain, by binding to, and partially blocking the transporter proteins that normally remove those monoamines from the synaptic cleft. However, considering the close similarities between ethylphenidate and methylphenidate and the fact that methylphenidate, like cocaine, actually does not primarily act as a "classical" reuptake inhibitor, but rather as an "inverse agonist at the DAT" (also called a "negative allosteric modulator at the DAT"), it is at least very likely that ethylphenidate also primarily acts as an inverse DAT agonist instead of (or at least only secondarily) as a classical reuptake inhibitor (which could be called a "competitive antagonist at the DAT" using a similar terminology as "negative allosteric modulator at the DAT", which per definition means that its mechanism is non-competitive). (en)
- L'éthylphénidate (EPH) est un psychostimulant et un produit proche du méthylphénidate. Les deux substances ont des effets pharmacologiques très similaires, au détail que l'éthylphénidate est plus sélectif des récepteurs dopaminergiques que le méthylphénidate. Ils possèdent des puissances similaires mais on remarque une différence sur l'activité de la norépinéphrine, elle serait plus faible et provoquerait donc moins de crises de paranoïa et de stress. Depuis mars 2015 ce NPS est interdit à la possession, vente et consommation en France. (fr)
- Etilfenidato (EPH) é uma droga psicoestimulante e um análogo próximo do metilfenidato. (pt)
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- 15765 (xsd:nonNegativeInteger)
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- Ethylphenidate-3D-ball-model.png (en)
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- -Ethyl 2-phenyl-2-piperidin-2-ylacetate (en)
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- Hepatic transesterification of prodrugs methylphenidate and ethanol (en)
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- Insufflation, vaporized, intravenous, intramuscular, rectal, oral, sublingual (en)
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- AIVSIRYZIBXTMM-UHFFFAOYSA-N (en)
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- إيثيل فينيدات هو منبّه ومشابه بنيوي قريب من ميثيل فينيدات. تقوم هذه المادة بدور مثبط استرداد للدوبامين وللنورإبينفرين، مما يرفع من تركيز هذه النواقل العصبية في الدماغ. يستقلب إيثيل فينيدات إلى ميثيل فينيدات ، وتتم العملية في الكبد عبر تفاعل . (ar)
- L'éthylphénidate (EPH) est un psychostimulant et un produit proche du méthylphénidate. Les deux substances ont des effets pharmacologiques très similaires, au détail que l'éthylphénidate est plus sélectif des récepteurs dopaminergiques que le méthylphénidate. Ils possèdent des puissances similaires mais on remarque une différence sur l'activité de la norépinéphrine, elle serait plus faible et provoquerait donc moins de crises de paranoïa et de stress. Depuis mars 2015 ce NPS est interdit à la possession, vente et consommation en France. (fr)
- Etilfenidato (EPH) é uma droga psicoestimulante e um análogo próximo do metilfenidato. (pt)
- Ethylphenidate (EPH), also known as Baxtercaine in the United Kingdom is a psychostimulant and a close analog of methylphenidate. Ethylphenidate acts as both a dopamine reuptake inhibitor and norepinephrine reuptake inhibitor, meaning it effectively boosts the levels of the norepinephrine and dopamine neurotransmitters in the brain, by binding to, and partially blocking the transporter proteins that normally remove those monoamines from the synaptic cleft. (en)
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- إيثيل فينيدات (ar)
- Ethylphenidate (en)
- Éthylphénidate (fr)
- Etilfenidato (pt)
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