Antimigraine Preparations

Name
Antimigraine Preparations
Accession Number
DBCAT002225
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
EletriptanA triptan used for the treatment of migraines.
MethysergideAn ergot alkaloid used for the prophylaxis of migraine and cluster headaches.
ZolmitriptanA member of the triptan class of 5-HT(1B/1D/1F) receptor agonist drugs used for the acute treatment of migraine with or without aura in adults.
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
LisurideFor the management of Parkinson's Disease
ErgotamineAn alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches.
AlmotriptanA 5-HT1B/1D receptor agonist used to treat migraines.
NaratriptanA 5-HT1B/1D receptor agonist used to treat migraines.
RizatriptanA triptan used to treat migraines with or without aura.
FrovatriptanA 5-HT1B/1D receptor agonist used to treat migraines.
PizotifenA serotonin and tryptamine antagonist indicated for migraine prophylaxis.
DimetotiazineDimetotiazine has considerable antiemetic & serotonin antagonistic action used mainly in allergic skin conditions.
OxetoroneNot Annotated
IprazochromeNot Annotated
FlumedroxoneNot Annotated
ClonidineAn alpha-2 adrenergic agonist used to treat hypertension and severe cancer pain, among other conditions, and to treat withdrawal symptoms from various substances. It is also used to aid in the diagnosis of pheochromocytoma and to prevent migraines.
SumatriptanA serotonin receptor agonist used to treat migraines and cluster headaches.
ErenumabA calcitonin-gene related peptide antagonist used to prevent migraines.
GalcanezumabA calcitonin-gene related peptide antagonist used to prevent migraines and treat cluster headaches.
UbrogepantAn oral CGRP antagonist used in the acute treatment of migraine with or without aura.
FremanezumabA humanized monoclonal antibody directed against human calcitonin-gene related peptide to prevent migraines.
RimegepantAn oral CGRP receptor antagonist used for the acute treatment of migraines with or without aura in adults.
EptinezumabA monoclonal antibody directed against CGRP infused every 3 months for the preventive treatment of migraine in adults.
ZavegepantA calcitonin gene-related peptide receptor antagonist indicated for the acute treatment of migraine with or without aura.
AtogepantAn oral CGRP antagonist used for the preventative therapy of episodic migraine headaches.
LasmiditanAn oral 5HT1F agonist used for the acute treatment of migraine headache with or without aura.
NaproxenAn NSAID used to treat rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, polyarticular juvenile idiopathic arthritis, tendinitis, bursitis, acute gout, primary dysmenorrhea, and mild to moderate pain.
Drugs & Drug Targets
DrugTargetType
Eletriptan5-hydroxytryptamine receptor 1Dtarget
Eletriptan5-hydroxytryptamine receptor 1Atarget
Eletriptan5-hydroxytryptamine receptor 1Ftarget
Eletriptan5-hydroxytryptamine receptor 1Btarget
EletriptanCytochrome P450 3A4enzyme
EletriptanCytochrome P450 2D6enzyme
EletriptanCytochrome P450 2C9enzyme
EletriptanCytochrome P450 2C19enzyme
EletriptanProstaglandin G/H synthase 1enzyme
EletriptanCytochrome P450 2A6enzyme
EletriptanATP-dependent translocase ABCB1transporter
Methysergide5-hydroxytryptamine receptor 2Atarget
Methysergide5-hydroxytryptamine receptor 1Atarget
Methysergide5-hydroxytryptamine receptor 7target
Methysergide5-hydroxytryptamine receptor 2Ctarget
Methysergide5-hydroxytryptamine receptor 2Btarget
Methysergide5-hydroxytryptamine receptor 1Btarget
Methysergide5-hydroxytryptamine receptor 1Ftarget
Methysergide5-hydroxytryptamine receptor 1Etarget
MethysergideCytochrome P450 3A4enzyme
Zolmitriptan5-hydroxytryptamine receptor 1Dtarget
Zolmitriptan5-hydroxytryptamine receptor 1Btarget
Zolmitriptan5-hydroxytryptamine receptor 1Ftarget
ZolmitriptanCytochrome P450 1A2enzyme
ZolmitriptanAmine oxidase [flavin-containing] Aenzyme
Zolmitriptan5-hydroxytryptamine receptor 1Atarget
ZolmitriptanATP-dependent translocase ABCB1transporter
Zolmitriptan5-hydroxytryptamine receptor 7target
Zolmitriptan5-hydroxytryptamine receptor 2Atarget
Zolmitriptan5-hydroxytryptamine receptor 2Btarget
Zolmitriptan5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
DihydroergotamineCytochrome P450 3A4enzyme
DihydroergotamineAlpha-2A adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineATP-dependent translocase ABCB1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineD(2) dopamine receptortarget
DihydroergotamineD(3) dopamine receptortarget
DihydroergotamineD(4) dopamine receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
DihydroergotamineBeta-3 adrenergic receptortarget
LisurideD(1A) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 1Atarget
LisurideD(2) dopamine receptortarget
LisurideAlpha-2A adrenergic receptortarget
LisurideAlpha-2B adrenergic receptortarget
LisurideAlpha-2C adrenergic receptortarget
LisurideD(3) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 1Dtarget
Lisuride5-hydroxytryptamine receptor 2Btarget
Lisuride5-hydroxytryptamine receptor 2Atarget
LisurideD(4) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 2Ctarget
LisurideD(1B) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 1Btarget
LisurideCytochrome P450 3A4enzyme
Lisuride5-hydroxytryptamine receptor 7target
ErgotamineAlpha-1A adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 1Dtarget
Ergotamine5-hydroxytryptamine receptor 1Btarget
Ergotamine5-hydroxytryptamine receptor 2Atarget
ErgotamineAlpha-2A adrenergic receptortarget
ErgotamineD(2) dopamine receptortarget
ErgotamineCytochrome P450 3A4enzyme
ErgotamineAlpha-1B adrenergic receptortarget
ErgotamineAlpha-1D adrenergic receptortarget
ErgotamineATP-dependent translocase ABCB1transporter
ErgotamineD(1) dopamine receptortarget
Ergotamine5-hydroxytryptamine receptor 1Atarget
Ergotamine5-hydroxytryptamine receptor 1Ftarget
Ergotamine5-hydroxytryptamine receptor 2Ctarget
Ergotamine5-hydroxytryptamine receptor 2Btarget
ErgotamineAlpha-2C adrenergic receptortarget
Almotriptan5-hydroxytryptamine receptor 1Dtarget
Almotriptan5-hydroxytryptamine receptor 1Btarget
AlmotriptanCytochrome P450 3A4enzyme
AlmotriptanCytochrome P450 2D6enzyme
AlmotriptanAmine oxidase [flavin-containing] Aenzyme
AlmotriptanFlavin-containing monooxygenase 3enzyme
AlmotriptanCytochrome P450 2C19enzyme
AlmotriptanCytochrome P450 2E1enzyme
AlmotriptanCytochrome P450 2C8enzyme
Naratriptan5-hydroxytryptamine receptor 1Dtarget
Naratriptan5-hydroxytryptamine receptor 1Btarget
Naratriptan5-hydroxytryptamine receptor 1Ftarget
Naratriptan5-hydroxytryptamine receptor 1Atarget
NaratriptanAmine oxidase [flavin-containing] Aenzyme
Rizatriptan5-hydroxytryptamine receptor 1Dtarget
Rizatriptan5-hydroxytryptamine receptor 1Btarget
Rizatriptan5-hydroxytryptamine receptor 1Ftarget
RizatriptanAmine oxidase [flavin-containing] Aenzyme
RizatriptanCytochrome P450 2D6enzyme
Rizatriptan5-hydroxytryptamine receptor 1Atarget
Rizatriptan5-hydroxytryptamine receptor 1Etarget
Rizatriptan5-hydroxytryptamine receptor 7target
Frovatriptan5-hydroxytryptamine receptor 1Dtarget
Frovatriptan5-hydroxytryptamine receptor 1Btarget
FrovatriptanCytochrome P450 1A2enzyme
PizotifenMuscarinic acetylcholine receptor M2target
PizotifenMuscarinic acetylcholine receptor M1target
PizotifenMuscarinic acetylcholine receptor M3target
Pizotifen5-hydroxytryptamine receptor 2Atarget
Pizotifen5-hydroxytryptamine receptor 2Btarget
Pizotifen5-hydroxytryptamine receptor 2Ctarget
PizotifenHistamine H1 receptortarget
Pizotifen5-hydroxytryptamine receptor 1Atarget
Pizotifen5-hydroxytryptamine receptor 1Btarget
PizotifenAlpha-1A adrenergic receptortarget
PizotifenAlpha-1B adrenergic receptortarget
PizotifenAlpha-1D adrenergic receptortarget
PizotifenAlpha-2A adrenergic receptortarget
PizotifenAlpha-2B adrenergic receptortarget
PizotifenAlpha-2C adrenergic receptortarget
PizotifenUDP-glucuronosyltransferase 2B10enzyme
ClonidineAlpha-2A adrenergic receptortarget
ClonidineCytochrome P450 2D6enzyme
ClonidineAlpha-2B adrenergic receptortarget
ClonidineAlpha-2C adrenergic receptortarget
ClonidineSolute carrier family 22 member 3transporter
ClonidineOrganic cation/carnitine transporter 2transporter
ClonidineSolute carrier family 22 member 4transporter
ClonidineCytochrome P450 1A2enzyme
ClonidineCytochrome P450 3A4enzyme
ClonidineCytochrome P450 1A1enzyme
ClonidineCytochrome P450 3A5enzyme
ClonidineAlpha-1A adrenergic receptortarget
ClonidineAlpha-1B adrenergic receptortarget
ClonidineAlpha-1D adrenergic receptortarget
ClonidineAlbumincarrier
ClonidineAmine oxidase [copper-containing] 3target
Sumatriptan5-hydroxytryptamine receptor 1Dtarget
Sumatriptan5-hydroxytryptamine receptor 1Btarget
Sumatriptan5-hydroxytryptamine receptor 1Ftarget
SumatriptanAmine oxidase [flavin-containing] Aenzyme
Sumatriptan5-hydroxytryptamine receptor 1Atarget
SumatriptanSolute carrier organic anion transporter family member 1A2transporter
SumatriptanATP-dependent translocase ABCB1transporter
SumatriptanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SumatriptanSolute carrier organic anion transporter family member 1B1transporter
ErenumabCalcitonin gene-related peptide type 1 receptortarget
GalcanezumabCalcitonin gene-related peptide 1target
GalcanezumabCalcitonin gene-related peptide 2target
UbrogepantATP-dependent translocase ABCB1transporter
UbrogepantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
UbrogepantCytochrome P450 3A4enzyme
UbrogepantCytochrome P450 2C8enzyme
UbrogepantCytochrome P450 2C9enzyme
UbrogepantCytochrome P450 2D6enzyme
UbrogepantCytochrome P450 2C19enzyme
UbrogepantAmine oxidase [flavin-containing] Aenzyme
UbrogepantUDP-glucuronosyltransferase 1A1enzyme
UbrogepantSolute carrier organic anion transporter family member 1B1transporter
UbrogepantSolute carrier organic anion transporter family member 1B3transporter
UbrogepantSolute carrier family 22 member 6transporter
UbrogepantSolute carrier family 22 member 2transporter
UbrogepantCalcitonin gene-related peptide type 1 receptortarget
FremanezumabCalcitonin gene-related peptide 1target
FremanezumabCalcitonin gene-related peptide 2target
RimegepantCalcitonin gene-related peptide type 1 receptortarget
RimegepantATP-dependent translocase ABCB1transporter
RimegepantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RimegepantSolute carrier organic anion transporter family member 1B1transporter
RimegepantOrganic anion transporter 3transporter
RimegepantSolute carrier organic anion transporter family member 1B3transporter
RimegepantSolute carrier family 22 member 2transporter
RimegepantMultidrug and toxin extrusion protein 1transporter
RimegepantCytochrome P450 3A4enzyme
RimegepantCytochrome P450 2C9enzyme
EptinezumabCalcitonin gene-related peptide 1target
EptinezumabCalcitonin gene-related peptide 2target
ZavegepantCalcitonin gene-related peptide type 1 receptortarget
ZavegepantCytochrome P450 3A4enzyme
ZavegepantCytochrome P450 2D6enzyme
ZavegepantSolute carrier organic anion transporter family member 1B3transporter
ZavegepantHepatic sodium/bile acid cotransportertransporter
ZavegepantATP-dependent translocase ABCB1transporter
ZavegepantMultidrug and toxin extrusion protein 1transporter
ZavegepantMultidrug and toxin extrusion protein 2transporter
AtogepantCalcitonin gene-related peptide type 1 receptortarget
AtogepantCytochrome P450 3A4enzyme
AtogepantSolute carrier organic anion transporter family member 1B1transporter
AtogepantSolute carrier organic anion transporter family member 1B3transporter
AtogepantSolute carrier family 22 member 6transporter
AtogepantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AtogepantATP-dependent translocase ABCB1transporter
AtogepantSolute carrier family 22 member 1transporter
AtogepantMultidrug and toxin extrusion protein 1transporter
Lasmiditan5-hydroxytryptamine receptor 1Ftarget
LasmiditanATP-dependent translocase ABCB1transporter
LasmiditanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LasmiditanSolute carrier family 22 member 1transporter
LasmiditanMultidrug and toxin extrusion protein 1transporter
LasmiditanMultidrug and toxin extrusion protein 2transporter
LasmiditanCytochrome P450 2D6enzyme
NaproxenProstaglandin G/H synthase 1target
NaproxenProstaglandin G/H synthase 2target
NaproxenAlbumincarrier
NaproxenCytochrome P450 2C9enzyme
NaproxenCytochrome P450 1A2enzyme
NaproxenSolute carrier organic anion transporter family member 1A2transporter
NaproxenSolute carrier family 22 member 6transporter
NaproxenCytochrome P450 2C8enzyme
NaproxenUDP-glucuronosyltransferase 2B7enzyme
NaproxenPeptostreptococcal albumin-binding proteintarget
NaproxenBile salt export pumptransporter
NaproxenATP-dependent translocase ABCB1transporter
NaproxenUDP-glucuronosyltransferase 1A3enzyme
NaproxenUDP-glucuronosyltransferase 1-6enzyme
NaproxenUDP-glucuronosyltransferase 1A7enzyme
NaproxenUDP-glucuronosyltransferase 1A8enzyme
NaproxenUDP-glucuronosyltransferase 1A9enzyme
NaproxenUDP-glucuronosyltransferase 1A10enzyme
NaproxenOrganic anion transporter 3transporter
NaproxenPancreatic triacylglycerol lipasetarget